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Preparation and one-step purification of mono-125I-angiotensin II for radioligand binding assays

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Abstract

A one-step purification of mono-125I-angiotensin II prepared by the chloramine T procedure is described. The purification is effected on a cellulose cation exchange column with isocratic elution by 50 mM sodium acetate, pH 5.0. The purity of the mono-125I-angiotensin II was determined by thin layer chromatography, high pressure liquid chromatography, enzymatic digestion, radioreceptor assay, and radioimmunoassay. Preparation and purification of mono-125I-angiotensin II by this procedure offers significant advantages over existing methods for its preparation in terms of purity, simplicity, efficiency, and cost.

Original languageEnglish
Pages (from-to)137-150
Number of pages14
JournalJournal of Pharmacological Methods
Volume11
Issue number2
DOIs
StatePublished - Apr 1984
Externally publishedYes

ASJC Scopus Subject Areas

  • Pharmacology

Keywords

  • Angiotensin II
  • Angiotensin II receptors
  • Cation exchange chromatography
  • mono-I-Angiotensin II
  • Preparation
  • Purification

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